Isoform-selective activity-based profiling of ERK signaling
Abstract
We report a novel chemical biology approach to study isoform-specific activity of extracellular signal-regulated kinases (ERKs), which are key regulators of signal transduction and emerging drug targets for oncology.
Document Details
- Document Type
- Pub Defense Publication
- Publication Date
- Jan 01, 2018
- Source ID
- 10.1039/c8sc00043c
Entities
People
- Caroline E. Franks
- Ku-lung Hsu
- Myungsun Shin
Organizations
- Congressionally Directed Medical Research Programs
- National Institute of General Medical Sciences
- National Institute on Drug Abuse
- United States Army
- University of Virginia
- Yusuf Hamied Department of Chemistry