19F-Tagged metal binding pharmacophores for NMR screening of metalloenzymes

Abstract

This study demonstrates the screening of a collection of twelve 19F-tagged metal-binding pharmacophores (MBPs) against the Zn(ii)-dependent metalloenzyme human carbonic anhydrase II (hCAII) by 19F NMR.

Document Details

Document Type
Pub Defense Publication
Publication Date
Jan 01, 2021
Source ID
10.1039/d1cc01231b

Entities

People

  • Alysia J. Kohlbrand
  • Hyeonglim Seo
  • Kathleen E Prosser
  • Mark Kalaj
  • Seth M Cohen

Organizations

  • Achievement Rewards for College Scientists Foundation
  • National Institute of Allergy and Infectious Diseases
  • Natural Sciences and Engineering Research Council
  • United States Army
  • University of California
  • Yusuf Hamied Department of Chemistry

Tags

Fields of Study

  • Chemistry

Readers

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