Structural determinants of TRPV4 inhibition and identification of new antagonists with antiviral activity

Abstract

The transient receptor potential vanilloid 4 (TRPV4) cation channel participates in multiple physiological processes and is also at the core of different diseases, making this channel an interesting pharmacological target with therapeutic potential. However, little is known about the structural elements governing its inhibition.

Document Details

Document Type
Pub Defense Publication
Publication Date
Oct 15, 2020
Source ID
10.1111/bph.15267

Entities

People

  • Fanny Rubio‐moscardo
  • Fernando González‐nilo
  • Gemma Pérez‐vilaró
  • Jonathan Canan
  • Juana Díez
  • Miguel A. Valverde
  • Pablo Doñate‐macian
  • Yorley Duarte

Organizations

  • Andrés Bello University
  • Ministry of Science of Spain
  • Pompeu Fabra University
  • United States Army Institute of Surgical Research
  • University of Valparaíso

Tags

Fields of Study

  • Chemistry

Readers

  • Cellular and Molecular Pathways of Apoptosis.
  • Immunology
  • Systems Analysis and Design