A cholecystokinin B receptor antagonist and cocaine interaction, phase I study

Abstract

RPR 102681, a cholecystokinin‐B antagonist, increased dopamine (DA) release and reduced cocaine self‐administration in animals. This pilot study sought to assess the safety and pharmacokinetics (PK) of co‐administration of RPR 102681 and cocaine, and to confirm the DA release mechanism of RPR 102681.

Document Details

Document Type
Pub Defense Publication
Publication Date
Jun 20, 2018
Source ID
10.1111/cns.12994

Entities

People

  • Ahmed Elkashef
  • Andrew Crabb
  • Dean F. Wong
  • Frank Vocci
  • James Robert Brašić
  • John Hilton
  • Jurij Mojsiak
  • Kimberly R. Warren
  • Louis R. Cantelina Jr
  • Nora Chiang
  • Roberta Kahn
  • Weiguo Ye
  • Yun Zhou

Organizations

  • Friends Research Institute
  • Johns Hopkins Bloomberg School of Public Health
  • Johns Hopkins University
  • Morgan State University
  • National Institute on Drug Abuse
  • Uniformed Services University of the Health Sciences

Tags

Readers

  • Molecular and Cellular Biochemistry
  • Neurodegenerative Parkinson's Disease and Rickettsial Disease handbook, including the data level of dopamine, BC, neurons, and PD.
  • Neurotoxicology