The brain microenvironment mediates resistance in luminal breast cancer to PI3K inhibition through HER3 activation

Abstract

The brain microenvironment triggers HER3-dependent de novo resistance to therapies targeting PI3K or HER2 in HER2-positive and/or PIK3CA -mutant breast cancer cells.

Document Details

Document Type
Pub Defense Publication
Publication Date
May 24, 2017
Source ID
10.1126/scitranslmed.aal4682

Entities

People

  • Alan Huang
  • Angela Tam
  • Bhushankumar Patel
  • C. Ryan Miller
  • Carey K. Anders
  • Carlos L Arteaga
  • Carlotta Costa
  • Christina Wong
  • Dai Fukumura
  • Dan G Duda
  • David P Kodack
  • Divya Bezwada
  • Elena Brachtel
  • Gino B. Ferraro
  • Jantima Tanboon
  • Jeffrey A. Engelman
  • Jonas Kloepper
  • Kamila Naxerova
  • Mark Badeaux
  • Marni B Siegel
  • Melinda E. Sanders
  • Mónica Valeria Estrada
  • Qing Sheng
  • Rakesh Jain
  • Rakesh R Ramjiawan
  • Ram C Shankaraiah
  • Rita Das
  • Robert Schlegel
  • Shom Goel
  • Vasileios Askoxylakis
  • Xiaolong Qi
  • Yongchul Song
  • Z. Alexander Cao

Organizations

  • German Research Foundation
  • Harvard Medical School
  • KWF Kankerbestrijding
  • National Cancer Institute
  • Susan G. Komen for the Cure
  • United States Department of Defense
  • University of North Carolina
  • Vanderbilt-Ingram Cancer Center

Tags

Fields of Study

  • Biology
  • Chemistry

Readers

  • Molecular Biology and Genetics