In Vitro and In Vivo Characterization of Tebipenem, an Orally Active Carbapenem, against Biothreat Pathogens

Abstract

Bacillus anthracis and Yersinia pestis , the causative pathogens for anthrax and plague, respectively, along with Burkholderia mallei and Burkholderia pseudomallei are potential bioterrorism threats. Tebipenem pivoxil hydrobromide (TBP HBr) (formerly SPR994) is an orally available prodrug of tebipenem, a carbapenem with activity versus multidrug-resistant (MDR) Gram-negative pathogens, including quinolone-resistant and extended-spectrum-β-lactamase-producing Enterobacterales .

Document Details

Document Type
Pub Defense Publication
Publication Date
Apr 19, 2021
Source ID
10.1128/aac.02385-20

Entities

People

  • Akash Jain
  • Christopher D. Kane
  • Denise Pfefferle
  • Gabriel T. Meister
  • Henry Heine
  • Lisa M. Pysz
  • M. Autumn Smiley
  • Michael J Pucci
  • Michael J. Hackett
  • Michael S. Anderson
  • Nicholas P. Clayton
  • Sanae Lembirik
  • Stephanie A. Halasohoris
  • Steven D. Zumbrun

Organizations

  • Battelle Memorial Institute
  • Biomedical Advanced Research and Development Authority
  • Defense Threat Reduction Agency
  • United States Army Medical Research Institute of Infectious Diseases
  • University of Florida

Tags

Fields of Study

  • Biology
  • Chemistry

Readers

  • Microbial Pathology
  • Neurotoxicology