Phase I/II Trial of Enzalutamide and Mifepristone, a Glucocorticoid Receptor Antagonist, for Metastatic Castration-Resistant Prostate Cancer

Abstract

Although androgen deprivation therapy (ADT) and androgen receptor (AR) signaling inhibitors are effective in metastatic prostate cancer, resistance occurs in most patients. This phase I/II trial assessed the safety, pharmacokinetic impact, and efficacy of the glucocorticoid receptor (GR) antagonist mifepristone in combination with enzalutamide for castration-resistant prostate cancer (CRPC).

Document Details

Document Type
Pub Defense Publication
Publication Date
Feb 02, 2022
Source ID
10.1158/1078-0432.ccr-21-4049

Entities

People

  • Amanda K L Anderson
  • Anthony V. Serritella
  • Daniel Shevrin
  • Elia Martinez
  • Elisabeth I Heath
  • James L Wade
  • Joseph Schonhoft
  • Russell Z. Szmulewitz
  • Theodore Karrison
  • Walter M. Stadler
  • Yen-Lin Chu

Organizations

  • Decatur Memorial Hospital
  • Epic Sciences
  • NorthShore University HealthSystem
  • United States Department of Defense
  • University of Chicago
  • Wayne State University

Tags

Fields of Study

  • Biology
  • Medicine

Readers

  • Prostate Cancer Biology.