TETRAHYDROCANNABINOLS. I. SYNTHESIS OF THE FOUR ISOMERS OF 2-(3,5-DIMETHOXYPHENYL)-3-METHYLOCTANE.
Abstract
The objective of this program was to obtain the eight individual isomers of a tetrahydrocannabinol for pharmacological evaluation. The previously unknown alpha-n-amyl-beta-methyl-3,5-dimethoxyhydrocinnamic acid (V) has been synthesized and separated into its erythro and threo isomers. These were resolved, then each converted in a three-step reaction sequence into the four stereoisomers of 2-(3,5-dimethoxyphenyl)-3-methyloctane (VII). The configurations of the VII isomers have been assigned by a conformational analysis of the infrared absorption spectra of the carbinols (VI) from which they are derived. (Author)
Document Details
- Document Type
- Technical Report
- Publication Date
- Oct 01, 1964
- Accession Number
- AD0354224
Entities
People
- C. Parker Ferguson
- Herbert S. Aaron
Organizations
- Edgewood Chemical Biological Center