STUDIES OF PYRIDOXAL-PENICILLAMINE ANTAGONISM IN THE HUMAN,

Abstract

The pyridoxal-L-penicillamine antagonism previously studied by others in lower animals has now been studied in man by means of urinary xanthurenic acid (XA) excretion levels. Subjects of the present study, all Chinese, included 21 normal individuals and 2 patients with Wilson's disease. The studies involved urinary XA determinations, with and without tryptophan-loading tests, and with varying dosage combinations of penicillamines and pyridoxine hydrochloride. It was found that urinary XA excretions remained normal after DL-penicillamine or DL-tryptophan alone but increased when the two were taken together; pyridoxine hydrochloride prevented the increase. No increases in urinary XA excretion occurred when Dpenicillamine or N-acetyl-DL-penicillamine were used in place of the DL-penicillamine during tryptophan loading. These results support the thesis that a pyridoxal-Lpenicillamine antagonism can operate in the human, both in normal individuals and in those with Wilson's disease.(Author)

Document Details

Document Type
Technical Report
Publication Date
May 28, 1964
Accession Number
AD0613760

Entities

People

  • Jun-bi Tu
  • R. Quentin Blackwell
  • William C. Cooper
  • Yu-hwa Chen

Tags

DTIC Thesaurus Topics

  • Biological Sciences
  • Chemical Compounds
  • Excretion
  • Pharmacology
  • Pyridoxines
  • Tryptophan

Readers

  • Electrochemical Surface Science
  • Molecular and Cellular Biology
  • Toxicology/Environmental Toxicology