Molecular Indicators of Castration-Resistant Prostate Cancer

Abstract

Metastatic prostate cancers are commonly treated by agents designed to suppress androgen receptor (AR) signaling mediated by the full-length AR (AR-FL). Why some patients progress rapidly after treatment while others benefit with prolonged remission is an unsolved question. We propose approaches to develop molecular indicators of response and resistance that will enable prediction (before therapy) or early detection (during therapy) of therapeutic benefit. We will test the hypothesis that AR splice variants (AR-Vs) are molecular indicators of castration-resistant prostate cancer (CRPC). During the funding period, we achieved major milestones by completing RNA sequencing of 55 clinical specimens and yielding data supporting the clinical importance of AR-V7, by establishing an association of AR-V7 with resistance to two current FDA-approved AR targeting therapies, and by demonstrating the feasibility of serial AR-V7 testing in men undergoing standard-of-care treatments for metastatic CRPC. We conclude that detection of AR-V7 predicts treatment outcome in men with metastatic castration resistant prostate cancer initiating AR-targeting therapies.

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Document Details

Document Type
Technical Report
Publication Date
Dec 01, 2015
Accession Number
AD1004093

Entities

People

  • Jun Luo

Organizations

  • Johns Hopkins University

Tags

DTIC Thesaurus Topics

  • Androgen Receptors
  • Chemical Reactions
  • Detection
  • Diseases And Disorders
  • Enzyme Inhibitors
  • Gene Expression
  • Health Services
  • Neoplasms
  • New England
  • Oncology
  • Prostate Cancer
  • Proteins
  • Regression Analysis
  • Rna Sequence Analysis
  • Standards
  • Statistical Analysis
  • X-Ray Computed Tomography

Fields of Study

  • Medicine

Readers

  • Oncology
  • Prostate Cancer Biology.