Epilepsy: The Role of the Super Family of Voltage Gated Ion Channels

Abstract

The superfamily of voltage gated ion channels is composed of channels regulating sodium, calcium or potassium entry into cells, regulated by alterations in the membrane potential. Dysregulation of members of this family often leads to the development of epilepsy. This review focuses on different mutations in this superfamily that are linked to the development of epilepsy and details the known mutations, the role of the specific mutated ion channel and the clinical consequences of each mutation. Disruption of voltage gated ion channel function can lead to increased excitability and contribute towards the development of epilepsy. The position of the mutation within the ion channel gene often influences the clinical presentation of symptoms, even for mutations within the same gene. A common feature of the superfamily of voltage gated ion channels is an alpha selective pore with augmentation by pore modifying protein subunits. Mutation of either the alpha pore or augmenting auxiliary proteins significantly alters ion channel function. An understanding of the molecular mechanisms of inherited epilepsy, will assist in establishing the etiology of all types of epilepsy and thus aid in the development of targeted therapeutics.

Open PDF

Document Details

Document Type
Technical Report
Publication Date
Feb 22, 2011
Accession Number
AD1013327

Entities

People

  • Edward L. Jones

Organizations

  • Uniformed Services University of the Health Sciences

Tags

DTIC Thesaurus Topics

  • Anticonvulsants
  • Brain
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Epilepsy
  • Genetics
  • Medical Personnel
  • Membrane Potentials
  • Neurology
  • Neurons
  • Neurosciences
  • Proteins
  • Seizures

Fields of Study

  • Biology
  • Medicine

Readers

  • Electrochemical Engineering/ Fuel Cell Technologies
  • Molecular Biology and Genetics
  • Neuroscience