Control of Colon Cancer Progression by the Colon Microbiome

Abstract

This Research Project was funded to define the roles of bacterial pathogen proteins which modify host proteins by post-translational modification. We have made great progress in accomplishing all of the AIMS of this project. The NF-B pathwayis most critical for immune defense against infection, thereby frequently targeted by bacterial virulence effectors. NleE, aneffector from EPEC and related enteric bacteria, is a SAM-dependent methyltransferase that blocks host NF-B-mediatedinflammation. We have solved the crystal structure of NleE-SAM complex, which reveals a methyltransferase fold differentfrom those of known methyltransferases. We further identify a new NleE substrate: ZRANB3, which has well defined roles inPCNA binding and remodeling of stalled replication forks at sites of DNA damage. NleE-catalyzed cysteine methylation of theZRANB3-NZF domain also abolishes its K63-linked ubiquitin chain-binding activity, a key modification of PCNA which initiatesrepair. Specific inactivation of the NZF domain in ZRANB3 by NleE, and hence its DNA repair functions suggests a novel andunexpected link between EPEC infection, virulence proteins and genome integrity. We have also discovered a new NleE substrate: ZRANB1/ Trabid1 , which contains three target zinc fingers and differentially methylates these three fingers tomodulate binding to mixed ubiquitin linked chains. Trabid1 functions in the NF-kB pathway in innate immunity like TAB2/3.

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Document Details

Document Type
Technical Report
Publication Date
Aug 01, 2015
Accession Number
AD1018895

Entities

People

  • Frank Iii J. Rauscher

Organizations

  • Wistar Institute

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Bacteria
  • Bacterial Infections
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Crystal Structure
  • Cysteine
  • Infection
  • Medical Personnel
  • Molecular Dynamics
  • Molecules
  • Pattern Recognition
  • Proteins
  • Wound Infections

Fields of Study

  • Biology

Readers

  • Microbial Pathology
  • Molecular Biology and Genetics
  • Molecular and genetic basis of cancer.

Technology Areas

  • Biotechnology