Arylimidamide Azole Combinations against Leishmaniasis

Abstract

In vitro IC50's were determined for seventeen newly synthesized compounds. Most compounds showed high therapeutic indexes by displaying strong in vitro efficacy against L. major and L. donovani parasites but low in vitro toxicity when tested in a macrophage cell line. During the fourth (and last year) of this grant no compounds were tested in the in vivo models of cutaneous leishmaniasis.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2018
Accession Number
AD1064683

Entities

People

  • Brian Vesely

Tags

DTIC Thesaurus Topics

  • Anti-Infective Agents
  • Antifungal Agents
  • Biology
  • Biomedical Research
  • Cell Line
  • Cells
  • Chemotherapy
  • Health Services
  • Infection
  • Leishmania
  • Leishmaniasis
  • Macrophages
  • Parasites
  • Parasitology
  • Toxicity
  • Validation

Fields of Study

  • Biology

Readers

  • Parasitology and Pharmacology of Malaria.