The Cytoplasm Translocation of the Androgen Receptor Cofactor p44 as a Target for Prostate Cancer Treatment

Abstract

The over-proliferation of prostate epithelial cell is the first critical step that leads to prostate tumorigenesis. We demonstrated that p44 cytoplasm localization associates with this growth process and is essential for growth of prostate epithelial and prostate cancer cells. The proposed research tested the feasibility to target this growth process for prostate cancer treatment. We report that inhibition of p44 cytoplasm translocation by identified compounds suppressed growth and progression of prostate tumors in both tumor xenografts and Pten gen knockout mouse model. These results provided a new paradigm and anew strategy for treatment of prostate cancer. In addition, we also found that the posttranslational modifications of p44 regulated its subcellular localization during rpostate tumorigenesis.

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Document Details

Document Type
Technical Report
Publication Date
Dec 01, 2019
Accession Number
AD1094754

Entities

People

  • Zhengxin Wang

Organizations

  • Clark Atlanta University

Tags

DTIC Thesaurus Topics

  • Androgen Receptors
  • Androgens
  • Biology
  • Biomedical Research
  • Cancer
  • Cells
  • Chemical Compounds
  • Chemistry
  • Cytoplasm
  • Epithelial Cells
  • Genes
  • Genetics
  • Hyperplasia
  • Neoplasms
  • Pcr Testing
  • Prostate
  • Prostate Cancer

Fields of Study

  • Biology
  • Medicine

Readers

  • Molecular Biology and Genetics
  • Prostate Cancer Biology.