MYCN Reprograms Neuroblastoma Metabolism

Abstract

Despite current aggressive regimens, the majority of patients with MYCN amplification die due to drug-resistant disease, and further intensification ofchemotherapy will not significantly improve this outcome. We propose an entirely novel strategy to oppose MYCN oncogenic function in NB: by blockingthe metabolic reprogramming driven by MYCN. Based on our data and the recent literature, our guiding hypotheses are that: a) lipid metabolism is requiredfor NB tumorigenesis, and b) targeting MYCN-driven lipogenesis will effectively block NB tumor growth. We have demonstrated that lipid metabolism is aselective metabolic dependency of MYCN-driven tumors. MYCN drives both fatty acid (FA) synthesis and FA uptake to maintain NB cell survival. TargetingFA uptake effectively blocks NB in vivo tumor growth.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 2020
Accession Number
AD1124982

Entities

People

  • Cristian Coarfa
  • Eveline Barbieri
  • Ling Tao
  • Mirthala M. Smith

Organizations

  • Baylor College of Medicine

Tags

DTIC Thesaurus Topics

  • Abstracts
  • Amplification
  • Biological Staining And Labeling
  • Biomedical Research
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemotherapy
  • Combination Therapy
  • Covid-19
  • Diseases And Disorders
  • Fatty Acids
  • Health Services
  • Inhibition
  • Inhibitors
  • Lipid Metabolism
  • Lipids
  • Medical Personnel
  • Metabolism
  • Neoplasms
  • Neuroblastoma
  • Small Molecules
  • Survival
  • Targeting
  • Therapy

Fields of Study

  • Medicine

Readers

  • Oncology
  • Prostate Cancer Biology.