MYCN Reprograms Neuroblastoma Metabolism

Abstract

Despite current aggressive regimens, the majority of patients with MYCN amplification die due to drug resistant disease, and further intensification of chemotherapy will not significantly improve this outcome. We propose an entirely novel strategy to oppose MYCN oncogenic function in NB: by blocking the metabolic reprogramming driven by MYCN. Based on our data and the recent literature, our guiding hypotheses are that: a) lipid metabolism is required for NB tumorigenesis, and b) targeting MYCN-driven lipogenesis will effectively block NB tumor growth. We have demonstrated that lipid metabolism is a selective metabolic dependency of MYCN-driven tumors. MYCN drives both fatty acid (FA) synthesis and FA uptake to maintain NB cell survival. Targeting FA uptake effectively blocks NB in vivo tumor growth.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2022
Accession Number
AD1201582

Entities

People

  • Eveline Barbieri

Organizations

  • Baylor College of Medicine

Tags

DTIC Thesaurus Topics

  • Abstracts
  • Biomedical Research
  • Carrier Proteins
  • Cell Physiological Processes
  • Cells
  • Diseases
  • Fatty Acids
  • Health Services
  • Inhibition
  • Inhibitors
  • Law
  • Lipid Metabolism
  • Lipids
  • Medical Personnel
  • Metabolism
  • Neoplasms
  • Neuroblastoma
  • Survival
  • Targeting
  • Therapy
  • Vulnerability

Fields of Study

  • Medicine

Readers

  • Cardiovascular Physiology
  • Molecular Biology and Genetics
  • Prostate Cancer Biology.