Targeting PARP Inhibitor Resistance
Abstract
Various inhibitors of poly(ADP-ribose) (PAR) polymerase (PARPi) have recently entered the clinic for the treatment of patients with ovarian cancers defective in homology-directed DNA repair, e.g. due to the loss of BRCA1/2 function. Despite the success of this approved novel therapy, drug resistance is a major clinical hurdle. The overall goal of this project is to target PARPi resistance in BRCA1/2-mutated high-grade serous ovarian cancer (HGS-OvCa), in order to optimize the use of PARPi and to develop new therapeutic approaches to overcome drug resistance.
Document Details
- Document Type
- Technical Report
- Publication Date
- Oct 01, 2023
- Accession Number
- AD1221329
Entities
People
- Intidhar Labidi-Galy
- Sven Rottenberg
Organizations
- University of Bern