1,2,4-Benzotriazine 1-Oxides as Antifolate-Antimalarials.

Abstract

This work was directed towards the preparation of 3-amino-7-substituted phenylsulfonyl-1,2,4-benzotriazine 1-oxides; a general route to this series was found. Two other desired series of compounds, 3-amino-7-substituted phenylthio-1,2,4-benzotriazine 1-oxides and 3-amino-7-substituted benzylamino-1,2,4-benzotriazine 1-oxides were not prepared, however, the reactions involved in their attempted preparation is summarized.

Document Details

Document Type
Technical Report
Publication Date
Oct 01, 1974
Accession Number
ADA006215

Entities

People

  • W. Wesley Parish
  • William D. Johnston

Tags

DTIC Thesaurus Topics

  • Anti-Infective Agents
  • Antimalarials
  • Enzyme Inhibitors
  • Pharmacologic Actions

Fields of Study

  • Chemistry

Readers

  • Organic Chemistry