The Cholinergic System and Nociception in the Primate: Interactions with Morphine.

Abstract

In experiment 1, the shock titration task was used to evaluate the antinociceptive properties of five different classes of cholinergic compounds in the Rhesus monkey. It was found that only scopolamine and high doses of physostigmine were effective in elevating the shock threshold. The apparent antinociceptive effect of physostigmine, however, was difficult to separate from its nonspecific behavioral depressant effect and was probably not related to an increase in cholinergic tone. Experiment 2 examined the interaction of morphine with arecoline, scopolamine, and physostigmine. Only scopolamine (0.05 and 0.1 mg/kg) and high doses of physostigmine (0.1 mg/kg) interacted with morphine in the shock titration paradigm. The multiplicative interaction of morphine with scopolamine was confirmed in experiment 3 over a wider range of doses. It was concluded that morphine and the cholinergic compounds produce antinociceptive effects through different mechanisms of the pain system.

Document Details

Document Type
Technical Report
Publication Date
May 01, 1975
Accession Number
ADA010665

Entities

People

  • Agu Pert

Tags

DTIC Thesaurus Topics

  • Arecoline
  • Diseases And Disorders
  • Memory Devices
  • Monkeys
  • Morphine
  • Nervous System Diseases
  • Neurologic Manifestations
  • Pain
  • Primates
  • Rhesus Monkeys
  • Signs And Symptoms
  • Symptoms And General Pathology
  • Titration

Fields of Study

  • Biology
  • Psychology

Readers

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  • Neurotrauma and Rehabilitation Medicine.
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