Studies in the Rat and Monkey on Absorption, Distribution, Metabolism, Excretion and Pharmacokinetics of WR-180,409.H3PO4.

Abstract

The search for new, more-effective antimalarial compounds is a continuing process due to the development of strains of malaria resistant to current therapy. As a part of an integrated effort to obtain information on the absorption, distribution, metabolism, excretion, and pharmacokinetics of investigational new drugs prior to clinical trial, the author undertook studies on WR-180,409.H3PO4 (Threo-a-(2-piperidyl)-2-trifluoromethyl-6-(4-trifluoromethylphenyl)-4-pyridine methanol phosphate).

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Document Details

Document Type
Technical Report
Publication Date
Apr 01, 1977
Accession Number
ADA039668

Entities

People

  • R. L. Furner

Organizations

  • Southern Research

Tags

DTIC Thesaurus Topics

  • Absorption
  • Adrenal Glands
  • Alcohols
  • Blood
  • Blood Cells
  • Body Fluids
  • Cells
  • Intestines
  • Large Intestine
  • Materials
  • Metabolism
  • Metabolites
  • Methanols
  • Pilot Studies
  • Rhesus Monkeys
  • Small Intestine
  • Tissues

Fields of Study

  • Medicine

Readers

  • Oncology
  • Parasitology and Pharmacology of Malaria.
  • Systems Analysis and Design