Synthetic Analogs of Phospholipid Metabolites as Antimalarials.

Abstract

Initial year's progress is described toward the synthesis of analogs of phospholipids and of their biosynthetic intermediates as possible antimalarials of a new type. Emphasis was placed on phosphonic and phosphinic acid analogs of lecithin, phosphatidic acid, cytidine diphosphate diglyceride, and cytidine diphosphate choline. Nine compounds were submitted of which one was a major target and three were secondary target compounds. None of the substances so far tested showed appreciable antimalarial activity. (Author)

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Document Details

Document Type
Technical Report
Publication Date
Sep 28, 1977
Accession Number
ADA046528

Entities

People

  • Arthur F. Rosenthal

Tags

DTIC Thesaurus Topics

  • Acetic Acid
  • Alcohols
  • Chemical Synthesis
  • Chemistry
  • Chromatography
  • Fungi
  • Gas Chromatography
  • Hydrogen
  • Iodine Compounds
  • Materials
  • Nitriles
  • Organic Chemistry
  • Organophosphorus Compounds
  • Phosphonic Acids

Fields of Study

  • Chemistry

Readers

  • Analytical Chemistry
  • Parasitology and Pharmacology of Malaria.
  • Prostate Cancer Biology.