Chemotherapy of 'Trypanosoma rhodesiense'.

Abstract

The test system described herein was developed specifically to evaluate the trypanosomicidal activity of large numbers of candidate compounds. Based on blood-induced Trypanosoma rhodesiense infections in mice, it performs as a primary screen or as a secondary screen and confirmatory test and gives precise quantitative evaluations of chemical compounds that demonstrate potentially useful therapeutic and/or prophylactic activity in T. rhodesiense infections. Consequently, it is also a helpful guideline in the synthesis of new active agents. These agents include: (1) chemicals structurally related to compounds of known value in the treatment or prevention of T. rhodesiense infections; (2) chemicals structurally unrelated to compounds of known value in the treatment or prevention of T. rhodesiense infections and; (3) structural analogues of compounds that have demonstrated activity in our screening procedure and represent novel chemical groups.

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Document Details

Document Type
Technical Report
Publication Date
May 31, 1974
Accession Number
ADA052299

Entities

People

  • Dora S. Rane

Organizations

  • University of Miami

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Analogs
  • Biomedical Research
  • Chemical Compounds
  • Chemistry
  • Chemotherapy
  • Contracts
  • Dilution
  • Diseases And Disorders
  • Infection
  • Research Facilities
  • Security
  • Standards
  • Test And Evaluation
  • Trypanosomiasis
  • Wound Infections

Fields of Study

  • Chemistry

Readers

  • Parasitology and Pharmacology of Malaria.
  • Systems Analysis and Design