Pharmacological Studies on Clostridial Neurotoxins.
Abstract
Experiments have been done that compare the actions of botulinum toxin type A, tetanus toxin, diphtheria toxin and beta-bungarotoxin on the cholinergic neuromuscular junction. All four toxins bind to tissues without producing adverse effects; each of the toxins has its own unique class of receptors. After tissue binding has occurred, botulinum toxin, tetanus toxin and diphtheria toxin are internalized; this process is antagonized by chloroquine, ammonium chloride and methylamine hydrochloride. Beta-Bungarotoxin is not internalized and is not antagonized by the drugs just listed. Diphtheria toxin acts intracellularly to ADP-ribosylate elongation factor 2. The intracellular actions of botulinum toxin and tetanus toxin have not been determined.
Document Details
- Document Type
- Technical Report
- Publication Date
- Aug 01, 1982
- Accession Number
- ADA118812
Entities
People
- Lance L. Simpson
Organizations
- Columbia University