Preparation and Purification of Multigram Quantities of TAX and SEX.

Abstract

This final report describes the multigram preparation and purification of l-acetylhexahydro-3,5-dinitro-l,3,5-triazine (TAX) and the feasibility of preparing, purifying, and analyzing multigram quantities of l-acetyloctahydro-3,5,7-trinitro-1,3,5,7-tetr azocine (SEX) needed for toxicological testing. TAX was prepared by nitrolysis of 1,3,5-triacetylhexahydro-1,3,5-triazine (TRAT) using a mixture of trifluoroacetic anhydride (TFAA) and 100% nitric acid. A continuous plug-flow reactor design was found to be a rapid, efficient, and safe method for the preparation of TAX in kilogram quantities. The crude TAX, contaminated with 25% to 30% RDX, was obtained analytically pure (99.9+%) by high-pressure liquid chromatography (HPLC) on silica gel using nitromethane as the eluent. SEX was prepared by nitrolysis of 1,5-diacetyloctahydro-3,7-dinitro-1,3,5,7-tetrazocine (DADN), using a mixture of 30% oleum and 100% nitric acid. Conditions for the preparation of the DADN/SEX/HMX mixture were optimized and the process can be conducted batchwise. Thus SEX could be provided in the quantities desired for subsequent purification.

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Document Details

Document Type
Technical Report
Publication Date
Dec 01, 1981
Accession Number
ADA122816

Entities

People

  • Bruce D. Deas
  • Clifford D. Bedford
  • Majorie M. Broussard
  • Maria A. Geigel

Organizations

  • SRI International

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Alcohols
  • Anhydrides
  • Biomedical Research
  • Chemical Synthesis
  • Chemistry
  • Chlorides
  • Chromatographs
  • Chromatography
  • Column Chromatography
  • Equations
  • Fluoropolymers
  • High Pressure
  • Infrared Spectra
  • Liquid Chromatography
  • Materials
  • Melting Point
  • Organic Chemistry

Fields of Study

  • Chemistry

Readers

  • Analytical Chemistry
  • Organic Chemistry