Effect of Perfluorodecanoic Acid on the Efflux of 2-Aminopurine from L5178Y Cells

Abstract

Transporters in the cell membrane of animal cells are susceptible to the action of toxic environmental agents. L5178Y mouse leukemia cells were treated with 150 micrograms/ml perfluorodecanoic acid (PFDA), a toxicant, in growth medium for 24 hr at 30 C. The PFDA-treated cells were transferred to fresh growth medium to demonstrate recovery of the capacity to transport a fluorescent purine, 2-aminopurine (AP). The membrane flux of AP was estimated with a high-speed kinetic assay. The cells were preloaded with 100 micrometers AP and rinsed twice in a cold buffer. The preloaded cells were resuspended in buffer at 21 C and AP flux was estimated continuously from the fluorescence emission of AP at 370 nm. At the beginning of the recovery period, AP efflux from PFDA-treated cells was markedly inhibited in comparison with the untreated controls. After 2 days at 37 C, the count of PFDA-treated cells doubled and the initial rate of AP efflux returned to approximately 60% of the controls. After 6 days at 30 C, the cell count increased 2.7-fold and AP efflux returned to approximately 60% of the controls. The results of experiments with untreated control cells show that the initial rate of AP efflux is proportional to the intracellular AP concentration.

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Document Details

Document Type
Technical Report
Publication Date
Sep 15, 1984
Accession Number
ADA148835

Entities

People

  • Paul W. Wigler

Organizations

  • University of Tennessee

Tags

DTIC Thesaurus Topics

  • Acids
  • Aminopurines
  • Blood
  • Cell Count
  • Cell Membrane
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Data Acquisition
  • Emission
  • Fluorescence
  • Inhibitors
  • Observation
  • Organic Chemistry
  • Pharmacology
  • Professional Associations
  • Uric Acid

Fields of Study

  • Biology

Readers

  • Aquatic Ecology
  • Mathematics or Statistics
  • Toxicology/Environmental Toxicology