Preclinical Toxicology of New Drugs.

Abstract

Preclinical toxicology studies of WR238605, Succinate and Pyridostigmine Bromide are being performed to assist the U.S. Army Medical R&D Command (USAMRDC) in its decision of whether or not to allow widespread clinical use of these agents. Subacute (28 day) toxicity studies of WR238605, Succinate, a potential antimalarial agent, were conducted in rats and dogs. Toxicity studies to define the reversibility of pyridostigmine-induced changes in the morphology of the neuromuscular junction were conducted in rats. Additionally, subacute (14 day) toxicity studies of pyridostigmine, a reversible anticholinesterase inhibitor, were conducted in rats and dogs. Results of these studies are detailed in individual study reports. Briefly, oral doses of WR238605, Succinate produced methemoglobin formation.

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Document Details

Document Type
Technical Report
Publication Date
Apr 04, 1986
Accession Number
ADA166877

Entities

People

  • J. G. Page

Organizations

  • Battelle Memorial Institute

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Blood
  • Body Weight
  • Chemical Synthesis
  • Chemistry
  • Clinical Trials
  • Enzyme Inhibitors
  • Gastrointestinal Diseases
  • Hemorrhage
  • Inhibitors
  • Intestinal Diseases
  • Laboratory Animals
  • Medical Personnel
  • Methemoglobin
  • Pyridostigmine Bromide
  • Tissues
  • United States

Fields of Study

  • Medicine

Readers

  • Cardiovascular Physiology
  • Neurotoxicology
  • Technical Research and Report Writing.