Synthesis of Potential Trypanocides

Abstract

This report describes the synthesis of new compounds for evaluation as antiparasitic agents. Most of the biological data pertain to activity against Trypanosoma rhodesiense but limited data pertaining to leishmania, filarius and plasmodium are also included. Biological data is included for compounds prepared in an earlier contract. The salts are derivatives of imidazole, pyridine, thiazole, benizimidazole and imidazo (1,2-a) pyridine. High levels of in vivo activity are reported for many of the compounds.

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Document Details

Document Type
Technical Report
Publication Date
Dec 01, 1987
Accession Number
ADA199129

Entities

People

  • Richard J. Sundberg

Organizations

  • University of Virginia

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • 1-Ring Heterocyclic Compounds
  • Alcohols
  • Aluminum Hydride
  • Amines
  • Chemotherapy
  • Classification
  • Cold Water
  • Contracts
  • Drug Abuse
  • Ethers
  • Hydrazines
  • Hydroxides
  • Infection
  • Precipitation
  • Security
  • Trypanosomiasis
  • Water

Fields of Study

  • Chemistry

Readers

  • Organic Chemistry
  • Parasitology and Pharmacology of Malaria.