Structure and Design of Multipotent Peptide Microbicides

Abstract

Defensin peptides, naturally occurring neutrophil antibiotics, were purified and characterized functionally and structurally. Functional differences in microbicidal potency and spectrum were correlated with structural features resolved by NMR and crystallographic methods. Protocols were established for synthesis and disulfide formation of natural defensins and synthetic congeners; we are currently investigating the latter by structural and functional characterization. Peptides, Structure-activity relationships, Synthesis, Microbicides, Antimicrobial peptides.

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Document Details

Document Type
Technical Report
Publication Date
Apr 19, 1990
Accession Number
ADA220995

Entities

People

  • Michael E. Selsted

Organizations

  • University of California, Los Angeles

Tags

DTIC Thesaurus Topics

  • Anti-Bacterial Agents
  • Anti-Infective Agents
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Command Control Communications
  • Contracts
  • Crystal Structure
  • Crystals
  • Membrane Lipids
  • Military Research
  • North America
  • Phagocytes
  • Plastic Explosives
  • Rodents
  • Spectra
  • Two Dimensional

Fields of Study

  • Chemistry

Readers

  • Molecular and Cellular Biochemistry