Effects of Trypanocidal Drugs on the Function of Trypanosomes

Abstract

The glycerophosphate oxidase system has been solubilized and partially purified using ubiquinol as an alternate electron donor and octyl glucoside as detergent. Some properties of the solubilized ubiquinol oxidase were investigated. 1) Once the holoenzyme had been in contact with the detergent, 2) glycerol-3-phosphate could no longer be used as substrate, 3) no matter whether the detergent was added during the assay or in the solubilization procedure. However, activity of the oxidase component could then be measured procedure. However, activity of the oxidase component could then be measured with ubiquinol analogs such as CoQ 1, with its isoprenoic side chain, 2,3- dimethoxy-5-methyl-6-nonyl-1,4-benzoquinone (NB) or 2,3-dimethoxy-5-methyl-6- decyl-1, 4-benzoquinone (DB) with their saturated straight chain alkyl groups. NB was preferentially used because it is more stable than CoQ 1, and can be synthesized easily. Keywords: Alpha-glycerophosphate oxidase, Ubiquinol oxidase, Cytochrome b, Maxicircle DNA.

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Document Details

Document Type
Technical Report
Publication Date
Jun 30, 1983
Accession Number
ADA221467

Entities

People

  • George C. Hill

Organizations

  • Colorado State University

Tags

DTIC Thesaurus Topics

  • Acids
  • Amino Acids
  • Animals
  • Cells
  • Cellular Structures
  • Central Nervous System
  • Chemistry
  • Domestic Animals
  • Enzymes
  • Genetic Code
  • Health Services
  • Metabolism
  • Mitochondria
  • Molecular Biology
  • Nervous System
  • Phosphodiesterases
  • Trypanosomiasis

Fields of Study

  • Biology
  • Chemistry

Readers

  • Analytical Chemistry
  • Electrochemical Surface Science
  • Parasitology and Pharmacology of Malaria.

Technology Areas

  • Microelectronics