Chemical Preparation Laboratory for IND Candidate Compounds

Abstract

During the reporting period seven compounds were synthesized and submitted to USAMRIID for testing. Most of these compounds were modified nucleosides derived from ribavirin, selenazole and formycin B, together with triazole heterocycles and an organic ester. Compounds which remain under investigation are a large-scale preparation of Ribavirin as well as the exploratory synthesis of dimethyl-ribavirin amidine and prodrug ester. Subject terms: Nucleosides; Triazoles; Heterocycles; Antivirals; RND Candidates; Prep synthesis; RAI.

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Document Details

Document Type
Technical Report
Publication Date
Feb 08, 1990
Accession Number
ADA221500

Entities

People

  • E. M. Schubert

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Acquired Immune Deficiency Syndrome
  • Alcohols
  • Anhydrides
  • Arbovirus Infections
  • Benzoic Acids
  • Biomedical Research
  • Chlorides
  • Dna Viruses
  • Ethers
  • Infectious Diseases
  • Medical Personnel
  • Nucleosides
  • Plastic Explosives
  • Rift Valley Fever
  • Rna Viruses
  • Sodium Compounds
  • Viruses

Fields of Study

  • Chemistry

Readers

  • Parasitology and Pharmacology of Malaria.
  • Systems Analysis and Design