Synthesis of Nucleoside Analogues with Potential Antiviral Activity against Negative Strand RNA Virus Targets

Abstract

The work described here is an attempt to synthesis nucleoside analogues which are targetted against the replicase of negative-strand viruses. Two lines of investigation have been attempted: (i) the synthesis of 5-vinyl substituted pyrimidine ribonucleosides and (ii) the synthesis of potential nucleotide pro-drugs. A series of compounds of type (i) have been synthesised and submitted for biological evaluation. Strategies for the synthesis of compounds of type (ii) have been developed but we have not had time to prepare sufficient suitable material for testing purposes. (js)

Open PDF

Document Details

Document Type
Technical Report
Publication Date
Nov 01, 1989
Accession Number
ADA229411

Entities

People

  • Richard T. Walker

Organizations

  • University of Birmingham

Tags

DTIC Thesaurus Topics

  • Animal Diseases
  • Antiviral Agents
  • Chemical Synthesis
  • Chemistry
  • Medical Personnel
  • Organic Chemistry
  • Viral Structures
  • Virus Diseases

Fields of Study

  • Chemistry

Readers

  • Parasitology and Pharmacology of Malaria.
  • Virology (or Medical Virology).