Characterization of Ligand-Induced Endocytosis of EGF - Receptors.

Abstract

We have made progress this year in engineering and using a cell line that is conditionally defective in receptor-mediated endocytosis to directly assess the role of endocytosis in controlling cellular responses to activated EGF-R. We find, not surprisingly, that cells defective in endocytosis show a stronger proliferative response to FGF than wt cells. Surprisingly, we find that some EGF-R signaling pathways, specifically the MAP kinase activation and EGF-R phosphorylation itself are reduced in mutant cells relative to wt cells. Thus, endocytosis plays a role in specifying EGF-R signaling events, not just in attenuating them. Given the importance of endocytosis in EGF-R signaling our discovery, that Rho-family GTPases which are activated in response to growth factors are negative regulators of receptor-mediated endocytosis, may have important implications or control of receptor signalling. Finally we have begun to examine the role of epsl5, a tyrosine kinase substrate of the EGF-R which binds constitutively to the AP2 endocytic coat proteins, on endocytosis of EGF-R using our in vitro assay.

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 1996
Accession Number
ADA314743

Entities

People

  • Christophe Lamaze
  • Sandra L. Schmid

Organizations

  • Scripps Research

Tags

DTIC Thesaurus Topics

  • Cell Line
  • Cell Physiological Processes
  • Cell-Free System
  • Cells
  • Chemistry
  • Cytoskeleton
  • Engineering
  • Growth Factors
  • Kinases
  • Materials
  • Peptide Growth Factors
  • Phosphorylation
  • Proteins
  • Regulations
  • Regulators
  • Substrates
  • Tyrosine

Fields of Study

  • Biology
  • Computer science

Readers

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