In Vivo Footprinting of the Progesterone Receptor Gene in Human Breast Cancer Cells

Abstract

We have used in vivo genomic footprinting to examine the interaction of proteins with the 5' flanking region of the progesterone receptor gene in human MCF-7 breast cancer cells. DMS footprinting of the PR gene demonstrates that Spisites in the A promoter are protected in the absence of hormone, but are more extensively protected in the presence of estrogen. In contrast, an adjacent ERE half site is not protected in the presence or in the absence of hormone. DNase I footprinting demonstrates that regions flanking the ERE/Sp1 sites are more extensively protected after estrogen treatment and that two antiestrogens elicit different footprinting patterns. While the partial agonist, 4-hydroxytamoxifen, produce a footprinting pattern that was similar to that of in vitro-cleaved, naked genomic DNA, the pure antagonist, ICI 182,780, produced a footprinting pattern that was distinct from all other footprints observed.

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Document Details

Document Type
Technical Report
Publication Date
Mar 01, 1998
Accession Number
ADA345418

Entities

People

  • Ann M. Nardulli

Organizations

  • University of Illinois Urbana–Champaign

Tags

DTIC Thesaurus Topics

  • Breast Cancer
  • Cells
  • Chemistry
  • Culture Techniques
  • Cultured Cells
  • Diseases And Disorders
  • Estrogens
  • Hormones
  • Laboratory Animals
  • Materials
  • Neoplasms
  • Polymerase Chain Reaction
  • Progesterone
  • Proteins
  • Recombinant Dna
  • Small Molecules
  • Tumor Cell Line

Fields of Study

  • Biology

Readers

  • Breast cancer cell signaling and growth regulation.
  • Molecular Genetics