Radioimmunotherapy of Metastatic Breast Cancer Using Radiolabeled Tumor Specific Antibodies

Abstract

Over the last four years we conducted and published a radioimaging trial using In-i ii Mx-DTPA huBrE-3 in patients with metastatic breast cancer. The results suggest that it is possible to administer therapeutic doses of Y-90 NX-DTPA huBrE-3 to patients. We are currently enrolling patients onto therapeutic trials of dose fractionated Y-90 NX-DTPA huBrE-3 to patients with metastatic breast cancer. We have also performed numerous preclinical experiments in the nude mouse human tumor xemograft model. We have demonstrated significant anti-tumor efficacy of combination continuous infusion topotecan and Y-90 MX-DTPA BrE-3. After tumors were allowed to grow for 21 days, the combination of 2OOu%i of 9OYttrium and 1 mg/m2 for 14 days via Alzet pump demonstrated complete tumor regression in 10 of 13 mice. As demonstrated in subsequent experiments, tumor response was specific to the BrE-3 antibody. This effect persisted with dose fractionation of antibody. In vivo studies demonstrated an increase in apoptosis and a decrease cell proliferation rate which was additive in the presence of topotecan and Y-90 MX-DTPA BrE-3. In our final year we continued these experiments using gemcitabine in a human pancreative cell xenograft nude mouse model and demonstrated significant activity of combination Y-90 MX-DTPA BrE-3 and gemcitabine.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 1998
Accession Number
ADA368409

Entities

People

  • Carolyn Wassweheit

Organizations

  • NYU Langone Health

Tags

DTIC Thesaurus Topics

  • Breast Cancer
  • Cell Physiological Processes
  • Chemical Synthesis
  • Chemistry
  • Health Services
  • Medical Personnel

Fields of Study

  • Biology
  • Medicine

Readers

  • Oncology (Cancer Research).