Prediction of Antichollintergic Drug Response Using a Thermoregulatory Exchange Index

Abstract

Among the drugs used for treatment of psychoses are those compounds which have a degree of anticholinergic action directly on eccrine sweat glands which disrupts thermoregulation. Atropine (a potent nerve agent antidote) reduces thermoregulatory sweating causing intense heat storage often leading to hyperpyrexia. A heat exchange analysis was carried out using a database of previous studies in our Institute in which saline and atropine (2 mg im) were injected in 14 healthy male subjects before and after heat acclimation. Subjects walked on a treadmill in hot-dry and hot-wet environments. A new effective temperature (ET*) was generated that can be implemented in any heat exchange evaluation utilizing biophysical and physiological data including mean skin temperature, rectal temperature, heart rate, metabolic activity, and skin evaporative heat loss. Heat acclimation reduced ET* by some 2.5 degrees C when compared with the unacclimated state after atropine injection. Heat acclimation thereby potentially lessens the hazards of heatstroke caused by exercise in the heat with atropine injection. Such a heat exchange model can be used to predict responses to other anticholinergic agents and has potential relevance applied in understanding psychotropic drug-related hyperthermia.

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Document Details

Document Type
Technical Report
Publication Date
Jan 01, 2000
Accession Number
ADA376680

Entities

People

  • Margaret A. Kolka
  • Richard R. Gonzalez

Organizations

  • United States Army Research Institute of Environmental Medicine

Tags

DTIC Thesaurus Topics

  • Acclimatization
  • Body Temperature
  • Body Weight
  • Health Services
  • Heart Rate
  • Heat Energy
  • Heat Loss
  • Heat Transfer
  • Heat Transfer Coefficients
  • Hyperthermia
  • Latent Heat
  • Mental Disorders
  • Psychiatry
  • Psychotropic Drugs
  • Sweating
  • Tranquilizing Agents
  • Vapor Pressure

Readers

  • Cardiovascular Physiology
  • Exercise and Sports Science.
  • Toxicology/Environmental Toxicology

Technology Areas

  • Biotechnology