C-MYC Protein-Protein and Protein-DNA Interactions: Targets for Therapeutic Intervention

Abstract

Basic-helix-loop-helix (bHLH) transcription factor proteins are involved in cell growth and differentiation, and the bHLH protein c-Myc has been implicated in breast cancer. We have determined that the sequence preference and specificity with which particular bHLH protein subclasses bind DNA are determined by binding conformations, which in turn are dictated by certain bHLH DNA binding region amino acids that are critical for protein function, but not for binding affinity. The data identify subtle effects on DNA binding that have important biological consequences, and reveal mechanisms by which different protein sub-family members can bind to different sites that share the CANNTG consensus. The zinc finger protein TTP is induced by many growth factors, and is required for regulation of TNFalpha expression.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 1999
Accession Number
ADA381686

Entities

People

  • T. K. Blackwell

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Biomedical And Dental Materials
  • Blood
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemistry
  • Dna Sequence Analysis
  • Embryos
  • Fungi
  • Genetics
  • Growth Factors
  • Lymphocytes
  • Medical Personnel
  • Polymeric Films
  • Proteins
  • Rna Stability

Fields of Study

  • Biology
  • Chemistry

Readers

  • Breast cancer cell signaling and growth regulation.
  • Molecular Genetics