Amplified Genes in Breast Cancer: Molecular Targets for Investigation and Therapy

Abstract

Our research focused on investigating acentric, autonomously replicating DNA containing amplified oncogenes (double minute chromosomes, DMs) as such structures occur in a significant fraction of human cancers. We proposed to develop methods to rapidly isolate and genotype DMs, to identify drugs to eliminate DMs, and to identify the mechanism(s) by which they are eliminated. We developed strategies to specifically tag DMs in living cells to enable analysis of their behavior during the cell cycle to enable us to ascertain differences between acentric structures and normal chromosomes to aid in the development of DM elimination reagents. We also devised and implemented novel cell labeling strategies to develop tumor models to determine how DM containing cells contribute to tumorigenesis, and to ascertain whether agents that effect DM elimination in vitro reduces tumor cell viability in vivo. Powerful new strategies and molecular tools were made available to the research community to enable sophisticated analyses of normal and abnormal chromosomes in cancer cells, and to allow studies of the relationship between genotype, phenotype and drug sensitivity in vivo.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 1999
Accession Number
ADA382811

Entities

People

  • Geoffrey M Wahl

Organizations

  • Salk Institute for Biological Studies

Tags

DTIC Thesaurus Topics

  • Antineoplastic Agents
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Chromosomes
  • Genetics
  • Health Services
  • Organic Chemistry
  • Proteins

Fields of Study

  • Biology

Readers

  • Civilian Systems Systems Program Capability Development and Upgrade Support Activity Expense and Pay Management.
  • Molecular and genetic basis of cancer.
  • Oncology (Cancer Research).