Erb-2/HER2 Oncogene in Breast Cancer: Does Bivalency of Growth Factors Drive Tumorigenicity Through Receptor Heterodimerization

Abstract

The HER2/ErbB-2 oncogenic protein contributes to virulence of human breast cancer and serves as a useful target for cancer immunotherapy. However, the exact mechanism underlying ErbB-2 function is still unknown. Our studies of the last year have concentrated on the widely accepted possibility that ErbB-2 acts as a direct receptor for a still unknown growth factor. By screening several potential candidates we found no known growth factor that fulfills the expected attributes of an ErbB-2 specific ligand. However, this search resulted in the identification of a novel growth factor, which we named Neuregulin-4, whose direct receptor is ErbB-4 (see publication 1). Systematic comparison of all of the known ligands of ErbB proteins, including three viral molecules, led us to conclude that ErbB-2 may not function as a direct receptor for a specific ligand. Instead, our studies imply that it acts as a shared co-receptor for many, if not all, ErbB ligands (See publication 2). This conclusion explains the tumorigenic action of ErbB-2 in terms of the cross-talk between the stroma and the epithelial tumor cells.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 1999
Accession Number
ADA382955

Entities

People

  • Yosef Yarden

Organizations

  • Weizmann Institute of Science

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Biomedical And Dental Materials
  • Blood
  • Breast Cancer
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Cellular Structures
  • Chemical Synthesis
  • Chemistry
  • Epithelial Cells
  • Growth Factors
  • Identification
  • Molecules
  • Neoplasms
  • Peptide Growth Factors
  • Proteins

Readers

  • Breast cancer cell signaling and growth regulation.
  • Theoretical Analysis.

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech