Syntheses of Diazadithiacrown Ethers Containing Two 8-Hydroxyquinoline Side Arms

Abstract

Ten new diazadithiacrown ethers containing two 8-hydroxyquinoline (HQ) sidearms attached through the HQ 7-positions and four new diazadithiacrown ethers containing two HQ sidearms attached through the HQ 2-positions have been prepared. Some of these new ligands also contain a hydroxymethyl substituent. The starting macrocyclic diazadithiacrown ethers were obtained by treatment of a bis(_-chloroamide) with the appropriate dimercaptan using K2CO3 as the base followed by reduction of the resulting macrocyclic dithiadiamide by BH3-THF or by NaBH4 in the presence of BF3-ether as a catalyst. HQ-containing ligands 23-32 were synthesized by a Mannich reaction of the secondary macrocyclic diamines with the substituted-8-hydroxyquinoline. HQ-containing ligands 33-36 were prepared by reductive amination of the secondary macrocyclic diamines with 8-hydroxyquinoline-2-carbaldehyde.

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Document Details

Document Type
Technical Report
Publication Date
Apr 17, 2001
Accession Number
ADA389135

Entities

People

  • G. P. Xue
  • H. C. Song
  • J. A. Chiara
  • J. S. Bradshaw
  • Y. W. Chen

Organizations

  • Brigham Young University

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DTIC Thesaurus Topics

  • Abstracts
  • Alkylating Agents
  • Biochemistry
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Crown Ethers
  • Ethers
  • Governments
  • Heavy Metals
  • Information Operations
  • Metals
  • Military Research
  • Organic Chemistry
  • United States
  • United States Government

Fields of Study

  • Chemistry

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