Functional Analysis of the ErbB4 Receptor Tyrosine Kinase

Abstract

This IDEA award is supporting our efforts to elucidate the roles that the ErbB4 receptor tyrosine kinase plays in breast cancer. We have generated three constitutively active mutants of ErbB4. Unlike constitutively active ErbB1 or ErbB2 mutants, the constitutively active ErbB4 mutants DO NOT couple to increased cell proliferation, to anchorage independent growth, or to a loss of contact inhibition in rodent fibroblast cell lines. Moreover, at least one of the constitutively active ErbB4 mutants is coupled to inhibition of colony formation in human mammary (tumor) cell lines and to inhibition of mammary (tumor) cell line proliferation. This suggests that ErbB4 is coupled to mammary tumor suppression in vivo.

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Document Details

Document Type
Technical Report
Publication Date
Jul 01, 2001
Accession Number
ADA396641

Entities

People

  • David J. Riese

Organizations

  • Purdue Research Foundation

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Biological Factors
  • Breast Cancer
  • Cancer
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Epithelial Cells
  • Genetics
  • Health Services
  • Organic Chemistry
  • Peptide Growth Factors
  • Peptides
  • Proteins

Fields of Study

  • Biology

Readers

  • Breast cancer cell signaling and growth regulation.