Mapping Critical DNA Sequence Elements Required for Amplification of erbB2 in Breast Cancer

Abstract

Recent studies show that 80-90% of breast carcinomas are associated with gene amplification. Each amplicon most likely has an origin of replication. In Drosophila, DmORC (Origin Recognition Complex) binds to specific DNA sequences and this binding is essential for chorion gene amplification. To study the implications of replication initiator proteins to gene amplification, we characterized two proteins required for DNA replication (ORC2 and Mcml0) . We created hypomorphic mutation in the ORC2 gene of a cancer cell line through homologous recombination. We found that these cells failed to support the replication of an extrachromosomal plasmid bearing the oriP replicator of Epstein Barr virus (EBV) . Geminin, an inhibitor of replication initiation complex, inhibited replication of this episome. The result identifies a novel means by which to cure cancer with gene amplification where the amplicons are carried as episomes. We also report that Xenopus Mcml0 (XMcml0) is not required for origin binding of XMcm2-7. Instead, the chromatin binding of XMcml0 at the onset of DNA replication requires chromatin-bound XMcm2-7, and it is independent of Cdk2 and Cdc7. In the absence of XMcml0, XCdc45 binding, XRPA binding, and initiation-dependent plasmid supercoiling are blocked. Therefore, XMcml0 performs its function after pre-RC assembly and before origin unwinding.

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Document Details

Document Type
Technical Report
Publication Date
May 01, 2002
Accession Number
ADA406150

Entities

People

  • Anindya Dutta
  • Yuichi Machida

Organizations

  • Brigham and Women's Hospital

Tags

DTIC Thesaurus Topics

  • Biomedical And Dental Materials
  • Breast Cancer
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Colon Cancer
  • Eukaryotes
  • Fungi
  • Genetics
  • Health Services
  • Polymer Chemistry
  • Polymeric Films
  • Proteins
  • Tumor Cell Line

Fields of Study

  • Biology

Readers

  • Molecular Biology and Genetics
  • Molecular Genetics