Interaction Between a Novel p21 Activated Kinase (PAK6) and Androgen Receptor in Prostate Cancer

Abstract

The androgen-signaling pathway is important for the growth and progression of prostate cancer. The cell cycle signaling regulated by mitogen activated protein/extracellular-signal-regulated kinase (MAPKIERK) have been linked to tumorigenesis. The p2l-activated kinases (PAKs) are members of a growing class of Rac/Cdc42-associated Ste20-like ser/thr protein kinases. Recent studies have shown that MAPK/ERK signaling can be mediated via Cdc42/Rac-stimulation of PAK activity. Recently, we demonstrated a specific interaction between a novel PAK protein, PAK6, and AR. This finding provided the first link between PAK-mediated signaling to the steroid hormone receptor pathway. In this study, we propose to assess the biological roles of PAK6 in prostate cancer cells, and to examine the expression of PAK6 in prostate tissues. We anticipate that by completing the objectives proposed in this grant, we will obtain fresh insight into the regulatory processes of AR and PAK6 that may be targeted for the development of a drug in the treatment of prostate cancer.

Open PDF

Document Details

Document Type
Technical Report
Publication Date
Feb 01, 2003
Accession Number
ADA415338

Entities

People

  • Zijie Sun

Organizations

  • Stanford University Medical Center

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Androgen Receptors
  • Cancer
  • Cell Membrane
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Cytoskeleton
  • Genetics
  • Hormones
  • Neoplasms
  • Prostate Cancer
  • Proteins
  • Tissues

Fields of Study

  • Biology

Readers

  • Cellular and Molecular Pathways of Apoptosis.
  • Oncology (Cancer Research).