Targeting of an Anti-Metastatic and Anti-Angiogenic Compound to Breast Tumors

Abstract

Our laboratory is studying anastellin, a fragment of fibronectin that inhibits angiogenesis, tumor growth and metastasis in vivo. By fusing anastellin with peptides that home to specific vascular sites in angiogenic vasculature, I am testing whether the concentration of anastellin at the angiogenic endothelium can be increased, and whether that would improve the anti-angiogenic activity of anastellin. I have found that targeting anastellin to angiogenic blood vessel endothelium in vivo does not improve the efficacy of anastellin. However, in contrast, targeting anastellin to lymphangiogenic vessels has a significant inhibiting effect on the development of lymphatic vasculature. These findings are interesting, because eliminating tumor lymphatics is a key step in inhibiting tumor metastasis.

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 2003
Accession Number
ADA417959

Entities

People

  • Maria Akerman

Organizations

  • Sanford Burnham Prebys Medical Discovery Institute

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Abstracts
  • Angiogenesis
  • Biomedical Research
  • Blood
  • Blood Vessels
  • Breast Cancer
  • Cancer
  • Cells
  • Contrast
  • Endothelial Cells
  • Endothelium
  • Lead Compounds
  • Lymphatic Vessels
  • Metastasis
  • Neoplasms
  • Targeting

Fields of Study

  • Biology
  • Medicine

Readers

  • Oncology (Cancer Research).
  • Parasitology and Pharmacology of Malaria.