Breast Tumor Kinase Signaling in Breast Cancer

Abstract

We previously demonstrated that the breast tumor kinase Brk can phosphorylate and inhibit the RNA-binding protein Sam68, which plays important roles in RNA metabolism associated with growth. Two novel Sam68-like mammalian proteins SLMl and SLM2 were identified, and cotransfection of NMuMG cells with different Brk expression constructs and either GFP-SLM1 or GFP-SLM2 revealed a direct correlation between Brk activity and the level of SLM1 and SLM2 phosphorylation. Mutation of the terminal tyrosine in Brk (Brk Y-F) increased the level of SLM protein phosphorylation. Localization of tyrosine phosphorylated proteins was examined in NMuMG cells cotransfected with Brk constructs and GFP-tagged substrates. Interestingly phosphotyrosine immunoreactivity was restricted to the nucleus and co-localized with the GFP-tagged nuclear substrates only when Brk Y-F was expressed. Expression of wild type Brk resulted in phosphorylation of cytoplasmic and nuclear proteins. This suggests a role for the carboxy terminal tyrosine in localization of Brk.

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 2003
Accession Number
ADA417996

Entities

People

  • Angela L. Tyner

Organizations

  • University of Illinois at Chicago

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Breast Cancer
  • Carrier Proteins
  • Cell Line
  • Cells
  • Confocal Microscopy
  • Department Of Defense
  • Epithelial Cells
  • Gene Expression
  • Mammary Glands
  • Mutations
  • Neoplasms
  • Phosphorylation
  • Proteins
  • Substrates
  • Terminals
  • Tyrosine

Fields of Study

  • Biology

Readers

  • Breast cancer cell signaling and growth regulation.
  • Molecular Genetics