Fundamental Patterns Underlying Neurotoxicity Revealed by DNA Microarray Expression Profiling

Abstract

The selective neurotoxins 1-methyl-4-phenylpyribinium (MPP+) and 6-hydroxydopamine (6-OHDA) have been widely used to generate animal models of Parkinson's disease (PD). To understand the genetic events associated with these neurotoxins, microarray technology served to monitor differences in gene expression patterns in normal versus pathological conditions. Microarray analysis of RNA isolated form toxin treated samples revealed that the stress induced transcription factor CHOP was dramatically up regulated by bothe toxins. 6-OHDA also induced a large number of genes involved in endoplasmic reticulum (ER) stress and unfolded protein response (UPR) such as ER chaperones and elements of the ubiquitin-proteasome system. RT-PCR, Western blotting, and immunocytochemical approaches were used to ouantify and temporarily order the UPR pathways involved in neurotoxin- induced cell death. 6-OHDA, but not MPP+, significantly increased hallmarks of UPR such as BiP, c-jun, and processed Xbpl mRNA. Both toxins increased the phosphorylation of UPR proteins, PERK and eTF2alpha, but only 6-OHDA increased phosphorylation of c-jun. Thus, 6-OHDA triggers multiple pathways associated with UPR, whereas MPP+ exhibits a more restricted response. 6-OHDA induced similar responses in primary dopaminergic neurons. These experiments will help clarify the molecular mechanisms associated with 6-OHDA and MPP+ toxicity and might aid in developing novel therapeutic avenues relevant to PD.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2003
Accession Number
ADA426087

Entities

People

  • Karen L. O'malley

Organizations

  • University of Washington

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Carrier Proteins
  • Cell Physiological Processes
  • Cells
  • Cellular Structures
  • Chemical Synthesis
  • Chemistry
  • Confocal Microscopy
  • Dna Microarrays
  • Endoplasmic Reticulum
  • Gene Expression
  • Health Services
  • Microarray Analysis
  • Neurons
  • Parkinson'S Disease
  • Proteins
  • Transcription Factors

Fields of Study

  • Biology

Readers

  • Molecular Biology and Genetics
  • Neurodegenerative Parkinson's Disease and Rickettsial Disease handbook, including the data level of dopamine, BC, neurons, and PD.

Technology Areas

  • Biotechnology