EGFR Activation by Spatially Restricted Ligands

Abstract

Misregulation of Transforming Growth Factor alpha (TGFalpha) and increased Epidermal Growth Factor Receptor (EGFR) activity has been associated with an increased prognosis of breast cancer (LeMaistre, 1994). TGFalpha and EGFR are required for normal breast development, but deregulation of this signaling pathway can result in uncontrolled proliferation and transformation (Matsui, 1990). 1 am studying the mechanism of TGFalpha activation of EGFR in the model organism Drosophila melanogaster in order to understand how post-transcriptional regulators of TGFalpha function to establish proper ligand expression. The purpose of this project is to identify factors that establish and maintain the tight localization of Gurken (Grk; a Drosophila TGFalpha-like ligand) that is necessary to produce spatially- restricted activation of the EGFR during ovary development (Schupbach, 1987; Neuman- Silberberg & Schupbach, 1993; 1994). These factors could define potential causes of EGFR misregulation, at the level of ligand production, that result in human breast cancer. I am integrating genetic and biochemical methods to study the effects of CG6554, Hrb27C, and Bruno on Grk expression. All three proteins interact with Squid (Sqd), a negative regulator of Grk (Kelly, 1993; Norvell et al. 1999).

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 2004
Accession Number
ADA426969

Entities

People

  • Jennifer S. Goodrich

Organizations

  • Princeton University

Tags

DTIC Thesaurus Topics

  • Breast Cancer
  • Carrier Proteins
  • Cells
  • Chemistry
  • Chromosome Structures
  • Chromosomes
  • Diptera
  • Genes
  • Genetic Structures
  • Genetics
  • Growth Factors
  • Health Services
  • Mrna
  • Neoplasms
  • Peptide Growth Factors
  • Proteins
  • Rodents

Readers

  • Breast cancer cell signaling and growth regulation.

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech