Targeting of an Anti-Metastatic and Anti-Angiogenic Compound to Breast Tumors

Abstract

This project concerns anastellin, a fragment of fibronectin that inhibits angiogenesis, tumor growth, and metastasis in vivo. It also concerns anginex, synthetic peptide with anti-angiogenic and anti-tumor effects. We have found that anginex resembles anastellin in several biochemical aspects, and that anginex, like anastellin, depends on circulating plasma fibronectin to be active in vivo. We have also found that anginex and anastellin in complex with fibronectin home to angigenic vasculature. It is possible that the fibronectin RGD sequence may function as the homing sequence of the peptide-fibronectin complexes to angiogenic endothelium in vivo.

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 2004
Accession Number
ADA427128

Entities

People

  • Maria Akerman

Organizations

  • Sanford Burnham Prebys Medical Discovery Institute

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Amino Acids
  • Anatomy
  • Angiogenesis
  • Biological Sciences
  • Biomedical Research
  • Blood
  • Blood Vessels
  • Breast Cancer
  • Cells
  • Diseases And Disorders
  • Electronic Mail
  • Endothelial Cells
  • Endothelium
  • Neoplasms
  • Sequences
  • Targeting

Fields of Study

  • Biology

Readers

  • Immunology
  • Molecular and Cellular Biochemistry
  • Oncology (Cancer Research).