Proteomic Analysis of Genistein Mammary Cancer Chemoprevention

Abstract

We have hypothesized that the phytoestrogen, genistein, exerts its chemopreventive actions by postnatally programming developmental modifications to genes/proteins that render the mammary gland less susceptible to cancer. The objective of this proposed research is to identify regulatory proteins responsible for conferring breast cancer protection. The specific aims are 1)to identify proteins that are differentially expressed in mammary glands of rats treated +/- the carcinogen, DMBA, and the chemopreventive agent, genistein, and 2) to collect proteins from interstitial fluid surrounding mammary glands of rats, and to identify and characterize the major proteins that are modulated by DMBA and genistein. Using 2-D gels and mass spectrometry, we have determined that GTP-cyclohyrolase 1, a protein that plays a prominent role in the production of tetrahydrobiopterin (BH4), is modulated by genistein. BH4 is an essential co-factor for the enzyme tyrosine hyroxylase. The latter is demonstrated to be up regulated at 50 days, but not at 21 days, hence, we postulate that tyrosine hydrolase expression is regulated via a programming mechanism. Up regulated tyrosine hydroxlase is associated with increased production of dopamine, the latter has been reported to inhibit angiogenesis. Aim 2 has been initiated.

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Document Details

Document Type
Technical Report
Publication Date
Jul 01, 2004
Accession Number
ADA428933

Entities

People

  • Coral A. Lamartiniere

Organizations

  • University of Alabama

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Breast Cancer
  • Cancer
  • Chemical Compounds
  • Chemistry
  • Dopamine
  • Drug Therapy
  • Glands
  • Mammary Glands
  • Mass Spectrometry
  • Neoplasms
  • Peptides
  • Production
  • Proteins
  • Proteomics
  • Two Dimensional
  • Tyrosine

Fields of Study

  • Biology

Readers

  • Molecular Biology and Genetics
  • Prostate Cancer Biology.

Technology Areas

  • Biotechnology