The Enzyme MnSOD Suppresses Malignant Breast Cell Growth by Preventing HIF-1 Activation

Abstract

Hypoxia inducible factor-1 (HIF-1) is a transcription factor that governs cellular responses to reduced O2 availability by mediating crucial homeostatic processes. The degradation of HIF-1 alpha subunit is redox regulated. Manganese superoxide dismutase (MnSOD) is an antioxidant enzyme that can modulate cellular redox environment. Here we show that MnSOD suppresses hypoxic accumulation of HIF-1 alpha protein. This suppression is biphasic depending on MnSOD activity. At low levels of MnSOD activity, HIF-1 alpha protein accumulates under hypoxic conditions in human breast carcinoma MCF-7 cells. At moderate levels of MnSOD activity (2-to 6-fold increase compared to parent cells), these accumulations are blocked. However, at higher levels of MnSOD activity (>6-fold increase), accumulation of HIF-1 alpha protein is again observed and the HIF-1 alpha protein level increases with increasing MnSOD activity. This biphasic modulation can be observed under both 1% O2 and 4% 02. Hypoxic induction of vascular endothelial growth factor (VEGF), a known HIF-1 targeted gene, is also suppressed by elevated MnSOD activity and its expression levels reflected the protein levels of HIF-1 alpha. These observations demonstrate that HIF-1 alpha accumulation is modulated not only by the levels of dioxygen but also the antioxidant enzyme MnSOD.

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Document Details

Document Type
Technical Report
Publication Date
May 01, 2004
Accession Number
ADA429516

Entities

People

  • Garry Buettner
  • Min Wang

Organizations

  • University of Iowa

Tags

DTIC Thesaurus Topics

  • Breast Cancer
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Endothelial Cells
  • Environment
  • Free Radicals
  • Growth Factors
  • Hypoxia
  • Modulation
  • Neoplasms
  • Oncology
  • Proteins
  • Regression Analysis
  • Tumor Cell Line

Readers

  • Molecular and Cellular Biochemistry
  • Naval Engineering and Maritime Security
  • Oncology (Cancer Research).