The Sensitivities of Yeast Strains Deficient in PDR ABC Transporters to Quinoline-Ring Antimalarial Drugs

Abstract

Data indicate a potential role for the Pdr5p P-glycoprotein ATP-binding-cassette (ABC) transporter in mediating chloroquine sensitivity in S. cervisae. This is consistent with the hypothesis that such a transporter plays a role in mediating quinoline-drug resistance in P. falciparum, and complements the results of previous studies on the parasite. Additional gene products also play a major role in mediating chloroquine sensitivity and resistance, apparently through the modulation of vacuolar pH in the parasite.

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Document Details

Document Type
Technical Report
Publication Date
Mar 12, 2004
Accession Number
ADA432795

Entities

People

  • Bradley C. Skillman
  • D. F. Wirth
  • H. Wolfger
  • K. Kuchler
  • Lyndal R. Emerson

Organizations

  • Walter Reed Army Institute of Research

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Anti-Infective Agents
  • Antimalarials
  • Cells
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Drug Resistance
  • Fungi
  • Genetics
  • Infectious Diseases
  • Parasites
  • Parasitology
  • Public Health
  • Quinolines
  • Resistance
  • Sensitivity
  • Tropical Medicine

Fields of Study

  • Biology

Readers

  • Molecular and Cellular Biochemistry
  • Parasitology and Pharmacology of Malaria.